Alisma

Alismataceae

Alisma plantago-aquatica

Also known as: Ze Xie, Water Plantain, Asian Water Plantain

Pregnancy B3
Lactation B3

clinical_notes Clinical Summary

Alisma (Alisma plantago-aquatica, Ze Xie) is a key diuretic herb in TCM, used for over two millennia to drain Dampness and promote urination in edema, dysuria, and hyperlipidemia.

Its protostane triterpenoids (alisol A/B and their acetates) confer diuretic, hypolipidemic, and hypoglycemic activity.

Human clinical trials support its use in cholesterol reduction and vertigo; concurrent use with diuretics or long-term high-dose use may risk electrolyte imbalance and nephrotoxicity.

Pregnancy Safety

B3

Traditional TCM restricts use in pregnancy due to draining nature; modern safety data are limited.

Lactation Safety

B3

Insufficient safety data during lactation; avoid.

warning Contraindications

  • Kidney Yin or Essence Deficiency with spermatorrhea (TCM) (caution)
    Theoretical
  • Long-term high-dose use (hepatotoxicity/nephrotoxicity risk) (caution)
    Theoretical
  • Fresh/raw root use (oral) (avoid)
    Theoretical
  • Concurrent diuretic or potassium-depleting medication (caution)
    Theoretical

vital_signs Clinical Profile

Primary Indications

  • check_circle edema
  • check_circle dysuria
  • check_circle urinary tract infection
  • check_circle hyperlipidemia
  • check_circle fatty liver
  • check_circle diarrhea
  • check_circle dizziness
  • check_circle vertigo
  • check_circle hypertension
  • check_circle kidney stones

Therapeutic Actions

diureticdamp-draininghypolipidemichypoglycemicanti-inflammatorynephroprotectivehepatoprotective

System Affinities

  • check_circle kidney
  • check_circle bladder
  • check_circle urinary

labs Active Constituents

alisol A

alisol B

alisol B 23-acetate

alisol A 24-acetate

alisol C 23-acetate

alismol

protostane triterpenoids

guaiane sesquiterpenes

polysaccharides

history_edu Traditional Use

Traditional Chinese Medicine (TCM)

Chinese Name

泽泻 (Zé Xiè)

Properties

Nature: cool

sweetbland
Meridians / Channels
KidneyBladder
TCM Indications
  • Damp-Heat
  • edema
  • dysuria
  • vertigo from phlegm-damp
  • hypertension
  • hyperlipidemia
Zang-Fu Organ Patterns
Damp-Heat in the BladderKidney Damp-HeatPhlegm-Damp Obstructing Clear YangKidney Yin Deficiency with Fire
Classical Formulas
Liu Wei Di Huang Wan (Six-Flavor Rehmannia Pill)Zhi Bai Di Huang WanZe Xie TangWu Ling San (Five Ingredient Powder with Poria)Jin Gui Shen Qi Wan
Notes

Chief diuretic herb in TCM. Dose-dependent actions: raw form is more draining, bran-fried form (fu chao) is gentler and used for Spleen support. Translates as 'Marsh Drain'.

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Traditional Uses Across Healing Systems

While many herbs lack controlled clinical trials, centuries of traditional practice across cultures provide valuable insight into their therapeutic applications.

TCM China
Listed in Shen Nong Ben Cao Jing (~200 AD); featured in Shang Han Lun Wu Ling San

Promotes urination and drains Dampness; clears Heat from the Kidneys and Bladder; resolves phlegm causing dizziness; regulates blood lipids. Core diuretic in the classic Liu Wei Di Huang Wan formula.

One of the most important damp-draining herbs in TCM. Classical texts note it can 'remove impure water' from the body.

Kampo Japan
Introduced from China

Known as Takusha; used in Hachimi-jio-gan, Rokumi-gan, and Gorei-san for edema, dysuria, and kidney-related vertigo.

Key component of multiple Kampo formulas.

Indigenous North America
Pre-colonial traditional use

Cherokee used Alisma subcordatum topically for wounds, bruises, and ulcers. Cree used the stem base for stomach and bowel conditions.

Different species but same genus with similar uses.

spa Parts Used

rhizome

Constituents
alisol Aalisol Balisol B 23-acetatealismolprotostane triterpenoidspolysaccharides
Indications
  • edema
  • dysuria
  • hyperlipidemia
  • vertigo
  • dizziness
Preparation

Rhizome harvested in winter; cleaned, sliced, and dried. Bran-fried (Fu Chao Ze Xie) form is gentler and used for Spleen deficiency diarrhea.

shield Safety

Contraindications — Evidence Basis

Kidney Yin or Essence Deficiency with spermatorrhea (TCM)
caution Theoretical

Traditional TCM contraindication; its draining, diuretic nature may deplete Yin/Jing.

Long-term high-dose use (hepatotoxicity/nephrotoxicity risk)
caution Theoretical

Long-term high-dose use or aqueous extracts at ≥50 g/kg in rats may cause tubular injury and hepatotoxicity via alisol A/B 23-acetate.

Fresh/raw root use (oral)
avoid Theoretical

Fresh roots and leaves contain toxic compounds that are deactivated by cooking/drying; use only dried or cooked preparations.

Concurrent diuretic or potassium-depleting medication
caution Theoretical

Additive diuretic effect may cause electrolyte imbalance, dehydration.

monitoring

Monitoring Parameters

Monitor during use, especially with prolonged or high-dose therapy.

Serum creatinine, BUN, and liver enzymes (ALT/AST)
Baseline and every 3 months with long-term use (>3 months)

Animal studies show potential renal tubular injury and hepatotoxicity with prolonged high-dose use.

flagThreshold: ALT/AST >2x ULN or creatinine increase >30% baseline: discontinue and reassess

Serum potassium and electrolytes
Baseline and at 4 weeks with concurrent diuretic use

Additive diuretic effect may cause hypokalemia or dehydration.

flagThreshold: Potassium <3.5 mEq/L: discontinue or adjust

menu_book Brinker F. Herbal Contraindications and Drug Interactions, 4th ed.

Toxicity

Toxic Dose

No acute toxicity at typical therapeutic doses (6–10 g dried rhizome). At 50 g/kg/day in rats, tubular toxicity observed.

Symptoms

Renal tubular injury, elevated liver enzymes with prolonged high-dose use.

Management

Discontinue; supportive care and monitoring of renal and hepatic function.

Adverse Effects

rare GI upsetelectrolyte imbalance (with prolonged use)dehydration

CYP Metabolism

Alisol compounds show potential induction of autophagy in renal cells; limited clinical interaction data.

swap_horiz Interactions

Spironolactone

Synergistic moderate

Class: Potassium-sparing diuretic

Mechanism

Alisma's triterpenoids increase urinary K+ excretion, but when combined with potassium-sparing diuretics the net effect on K+ is unpredictable. Additive diuresis raises the risk of dehydration and hyponatremia.

Clinical Guidance

Monitor electrolytes (especially K+) and volume status. Avoid combination in patients with advanced kidney or cardiac disease.

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Evidence Source Tian T, et al. Traditional uses, phytochemistry, pharmacology, toxicology and quality control of Alisma orientale. J Ethnopharmacol. 2014;158:373-387 View source open_in_new

Furosemide

Synergistic moderate

Class: Loop diuretic

Mechanism

Alisma triterpenes (alisol A, alisol B, alisol B 23-acetate) produce a dose-dependent diuretic effect by increasing urinary Na+, K+, and Cl- excretion and reducing aquaporin-2 mRNA in renal medullary cells. Additive diuresis with loop diuretics may lead to electrolyte depletion and dehydration.

Clinical Guidance

Monitor serum electrolytes (K+, Na+, Mg2+) and renal function. Adjust diuretic dose if volume depletion develops.

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Evidence Source Zhang X, et al. Diuretic activity of compatible triterpene components of Alismatis rhizoma. Molecules. 2017;22(9):1459 View source open_in_new

Lithium

Increased Effect high

Class: Mood stabilizer

Mechanism

Alisma's marked diuretic effect may alter renal lithium clearance and sodium balance, potentially raising serum lithium levels to toxic ranges, consistent with other strongly diuretic herbs.

Clinical Guidance

Avoid combination unless lithium levels and renal function are monitored closely. Watch for toxicity (tremor, confusion, ataxia).

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Evidence Source Tian T, et al. Traditional uses, phytochemistry, pharmacology, toxicology and quality control of Alisma orientale. J Ethnopharmacol. 2014;158:373-387 View source open_in_new

Atorvastatin

Synergistic low

Class: HMG-CoA reductase inhibitor (statin)

Mechanism

Alisma and its triterpenoids (especially alisol B 23-acetate) have well-documented hypolipidemic activity via modulation of lipid metabolism; combination with statins produces additive LDL lowering.

Clinical Guidance

Combination is generally beneficial. Monitor lipid panel routinely.

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Evidence Source Shu Z, et al. Alisma orientale: Ethnopharmacology, phytochemistry and pharmacology of an important traditional Chinese medicine. Am J Chin Med. 2016;44(2):227-251 View source open_in_new

Metformin

Synergistic low

Class: Biguanide antidiabetic

Mechanism

Alisma has demonstrated hypoglycemic activity via AMPK activation and improved insulin sensitivity in preclinical models; effects are complementary to metformin's mechanism.

Clinical Guidance

Monitor blood glucose. Dose adjustment rarely required; watch for hypoglycemia in tightly controlled patients.

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Evidence Source Lau CH, et al. Hypoglycemic activity of Alisma orientale. Phytomedicine 2008 View source open_in_new

Ibuprofen

Caution moderate

Class: NSAID

Mechanism

Both alisma and NSAIDs can affect renal hemodynamics; NSAIDs decrease renal prostaglandins while alisma's diuretic activity may exacerbate volume depletion, increasing risk of prerenal acute kidney injury when used together, especially in older adults.

Clinical Guidance

Avoid long-term concomitant use in patients with CKD or dehydration. Ensure adequate hydration and monitor renal function.

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Evidence Source Tian T, et al. Traditional uses, phytochemistry, pharmacology, toxicology and quality control of Alisma orientale. J Ethnopharmacol. 2014;158:373-387 View source open_in_new

Digoxin

Caution high

Class: Cardiac glycoside

Mechanism

Alisma-induced diuresis and potassium loss can precipitate digoxin toxicity; hypokalemia sensitizes myocardium to digoxin effects, increasing arrhythmia risk.

Clinical Guidance

Monitor serum potassium and digoxin levels. Replace potassium if depleted. Avoid combination in elderly patients with heart failure unless tightly monitored.

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Evidence Source Tian T, et al. Traditional uses, phytochemistry, pharmacology, toxicology and quality control of Alisma orientale. J Ethnopharmacol. 2014;158:373-387 View source open_in_new

hub Combinations

info

Synergistic pairings can enhance therapeutic outcomes, while knowing suitable substitutes helps when specific herbs are unavailable or contraindicated.

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Classical Formulas

2
Atractylodes
Traditional Use
Rationale

Used together in Ze Xie Tang for phlegm-damp vertigo and dizziness.

Clinical Evidence

Classical formula from Jin Gui Yao Lue.

link Jin Gui Yao Lue
Rehmannia
Strong Evidence
Rationale

Core pairing in Liu Wei Di Huang Wan — Ze Xie drains turbid water while Rehmannia nourishes Kidney Yin.

Clinical Evidence

Classic formula in wide use; extensively studied in hypertension, diabetes, and menopause.

link Bensky Formulas & Strategies, 2nd ed.
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Synergistic Combinations

2
Poria
Traditional Use
Rationale

Both drain dampness via urination; core pairing in Wu Ling San for water metabolism disorders.

Clinical Evidence

Classical Shang Han Lun formula.

link Shang Han Lun
Zhu Ling
Traditional Use
Rationale

Combined in Wu Ling San and Zhu Ling Tang to drain dampness and resolve heat without injuring Yin.

Clinical Evidence

Classic TCM pairing for urinary damp-heat.

link Shang Han Lun; Jin Gui Yao Lue

science Studies

search

Effects and potential mechanisms of Alismatis Rhizoma extracts on glucose and lipid metabolism: A systematic review and meta-analysis of rodent studies

Meta-Analysis
2025 |Authors. J Ethnopharmacol. 2025; PMID:40825387

This systematic review and meta-analysis of 29 preclinical rodent studies evaluated the efficacy and mechanisms of Alisma plantago-aquatica rhizome (AR) extracts on glucose and lipid metabolism disorders. AR extracts significantly improved fasting plasma glucose, postprandial glucose, insulin resistance (HOMA-IR), total cholesterol, triglycerides, LDL-C, and body weight in rodent models. Proposed mechanisms include antioxidant effects, anti-inflammatory activity, inhibition of gluconeogenesis, enhancement of insulin signaling, promotion of autophagy, and anti-fibrotic effects. Study quality was assessed by SYRCLE risk-of-bias tool, and statistical analysis followed CHSRI standards. The authors noted that while preclinical evidence is robust and consistent, well-designed human trials are still needed to translate these findings into clinical recommendations.

Cardiovascular HealthDiabetes Support
antidiabetichypolipidemicantioxidantinsulin sensitizationanti-inflammatory
View source open_in_new

Alisma plantago-aquatica polysaccharides ameliorate acetaminophen-induced acute liver injury by regulating hepatic metabolic profiles and modulating gut microbiota

In Vivo
2024 |Authors. Phytomedicine. 2024; PMID:39631232

This in vivo study investigated the hepatoprotective effects of Alisma plantago-aquatica polysaccharides (ARP50 and ARP70) in an acetaminophen (APAP)-induced acute liver failure mouse model. In vitro free radical scavenging assays confirmed notable antioxidant activity of both ARP fractions. In vivo, both polysaccharide fractions exerted dose-dependent protective effects against APAP-induced liver injury, with hepatic metabolite profiling revealing restoration of the liver antioxidant system through modulation of metabolism pathways. Gut microbiota analysis showed significant alterations associated with liver protection, suggesting a gut-liver axis mechanism. These findings provide first-in-kind evidence that Alisma polysaccharides protect against drug-induced acute liver injury through antioxidant and microbiota-modulating mechanisms.

Liver Health
hepatoprotectiveantioxidantgut microbiota modulationanti-inflammatory
View source open_in_new

medication Dosing

decoction

Dose Range

6–10 g dried rhizome

Frequency

1–2x/day

Notes

Classical TCM dose; decoct 20–30 minutes.

powder

Dose Range

1.5–3 g powdered rhizome

Frequency

2–3x/day

Notes

May be stirred into warm water or decoction.

menu_book
Reference Bensky Materia Medica, 3rd ed.

tincture

Dose Range

2–4 mL (1:5, 45% ethanol)

Frequency

2–3x/day

Notes

Modern Western herbal application; use only dried root to ensure safety.

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Reference Mills & Bone, Principles and Practice of Phytotherapy
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Disclaimer: This information is largely AI-generated and reviewed by human experts at Evara Health. It is intended for educational and clinical reference purposes only and should not replace professional medical advice.

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