Chinese Rhubarb

Polygonaceae

Rheum palmatum

Also known as: Da Huang, Turkey Rhubarb, Medicinal Rhubarb

Pregnancy D
Lactation C

clinical_notes Clinical Summary

Chinese Rhubarb (Rheum palmatum, Da Huang) is a classic purgative and blood-mover used in both Chinese medicine and Western pharmacopoeia.

At low doses it acts as a bitter astringent and digestive tonic; at higher doses its anthraquinones (sennosides, rhein, emodin) stimulate colonic peristalsis and drain 'heat accumulation.' Use is limited to short courses — ideally under 1-2 weeks — and contraindicated in pregnancy, lactation, intestinal obstruction, and chronic constipation from atonic or inflammatory causes.

Pregnancy Safety

D

Contraindicated due to pelvic-congesting and uterine-stimulant activity of stimulant anthraquinones.

Lactation Safety

C

Avoid; small amounts of anthraquinone metabolites may pass to milk and cause infant diarrhea.

warning Contraindications

  • Pregnancy (contraindicated)
    Theoretical
  • Lactation (avoid)
    Theoretical
  • Children <12 y (contraindicated)
    Theoretical
  • Intestinal obstruction / ileus / undiagnosed acute abdomen (contraindicated)
    Theoretical
  • Inflammatory bowel disease (Crohn's, UC) (avoid)
    Theoretical
  • Chronic stimulant-laxative use (>1-2 weeks) (caution)
    Clinically Proven
  • History of kidney stones / hyperoxaluria (caution)
    Theoretical
  • Concurrent digoxin, loop/thiazide diuretics, or corticosteroids (caution)
    Clinically Proven

vital_signs Clinical Profile

Primary Indications

  • check_circle Acute constipation with heat
  • check_circle Impacted bowel with abdominal distention
  • check_circle Acute appendicitis (as adjunct)
  • check_circle Cholestasis / jaundice
  • check_circle Upper GI bleeding (charred form)
  • check_circle Amenorrhea from Blood stasis
  • check_circle Burns (topical)

Therapeutic Actions

laxative (stimulant)purgative (high dose)cholagoguehemostatic (paradoxically, at low dose / charred)antimicrobialanti-inflammatoryastringent (at low dose)

System Affinities

  • check_circle gastrointestinal tract
  • check_circle hepatobiliary system
  • check_circle blood

labs Active Constituents

Anthraquinone glycosides

Tannins

Stilbenes

Resins

Calcium oxalate crystals

history_edu Traditional Use

Traditional Chinese Medicine (TCM)

Chinese Name

大黄 (Dà Huáng)

Properties

Nature: cold

bitter
Meridians / Channels
StomachLarge IntestineSpleenLiverHeart
TCM Indications
  • Heat accumulation with constipation
  • Damp-Heat jaundice
  • Blood stasis (amenorrhea, fixed masses)
  • Fire toxin with sores
  • Blood heat hemorrhage (charred form)
  • Yangming organ pattern (high fever, constipation, delirium)
Zang-Fu Organ Patterns
Stomach/Intestine Heat AccumulationLiver-Gallbladder Damp-HeatBlood StasisFire Toxin
Classical Formulas
Da Cheng Qi Tang (Major Order the Qi Decoction)Tao He Cheng Qi Tang (Peach Pit Decoction)Da Huang Mu Dan Tang (for appendicitis)Wen Pi TangSan Huang Xie Xin Tang
Notes

Processed forms differ: raw Da Huang is strongest purgative; wine-fried moves upward/blood; charred Da Huang (Da Huang Tan) is hemostatic. Cornerstone of Zhang Zhongjing's Yangming purgative strategy.

auto_stories

Traditional Uses Across Healing Systems

While many herbs lack controlled clinical trials, centuries of traditional practice across cultures provide valuable insight into their therapeutic applications.

TCM China
Documented in Shennong Ben Cao Jing (~200 BCE); foundational in Shang Han Lun (~220 CE)

Purges Heat and accumulation, drains Fire, cools Blood, invigorates Blood, expels Blood stasis, clears Damp-Heat.

One of the 'fifty fundamental herbs' in TCM.

Western Herbal Europe
Imported along Silk Road from ~9th century; pharmacopoeial in Europe from Medieval times

Used as bitter digestive tonic at low dose; as stimulant laxative for constipation at higher dose.

Turkey Rhubarb was historically a major trade commodity, more valuable than gold at times.

Unani Persia / Middle East
Used in Unani medicine since medieval period

Classified as hot-dry; used to purge 'burnt' humors and for jaundice.

Called 'Rawand Chini' in Unani pharmacopoeia.

spa Parts Used

root and rhizome

Constituents
Sennosides A-FRheinEmodinAloe-emodinChrysophanolTannins
Indications
  • Constipation
  • Heat accumulation
  • Jaundice
  • Upper GI bleeding (charred)
Preparation

Harvested in autumn from plants 3-5 years old. Sliced and dried. Processed forms: raw (strongest purgative), wine-fried (moves blood), charred (hemostatic), and steamed (gentler).

shield Safety

Contraindications — Evidence Basis

Pregnancy
contraindicated Theoretical

Stimulant anthraquinones cause pelvic congestion and may stimulate the uterus.

Lactation
avoid Theoretical

Anthraquinone metabolites may transfer to milk and cause infant diarrhea.

Children <12 y
contraindicated Theoretical

EMA: not recommended under 12 due to laxative risks.

Intestinal obstruction / ileus / undiagnosed acute abdomen
contraindicated Theoretical

Stimulant laxatives contraindicated in obstruction.

Inflammatory bowel disease (Crohn's, UC)
avoid Theoretical

Stimulant action may exacerbate mucosal inflammation.

menu_book Mills & Bone. Principles and Practice of Phytotherapy, 2nd ed. 2013
Chronic stimulant-laxative use (>1-2 weeks)
caution Clinically Proven

Associated with electrolyte depletion (hypokalemia), melanosis coli, and laxative dependence.

History of kidney stones / hyperoxaluria
caution Theoretical

High oxalate content may aggravate oxalate stone risk.

menu_book Clinical consensus
Concurrent digoxin, loop/thiazide diuretics, or corticosteroids
caution Clinically Proven

Hypokalemia from chronic stimulant laxatives potentiates digoxin toxicity.

monitoring

Monitoring Parameters

Monitor during use, especially with prolonged or high-dose therapy.

Serum potassium
Baseline and periodically with use >1 week

Chronic stimulant laxatives cause hypokalemia.

flagThreshold: K+ <3.5 mmol/L: discontinue and supplement.

Bowel frequency and stool consistency
Daily during acute use

Titrate to softest stool; avoid watery diarrhea.

flagThreshold: More than 2 loose stools/day: reduce dose.

Toxicity

Toxic Dose

At >1 g/day of anthraquinone-standardized extract for extended periods, electrolyte imbalance and laxative dependence develop. Acute overdose causes severe watery diarrhea.

Symptoms

Abdominal cramps, severe diarrhea, dehydration, hypokalemia, muscle weakness, arrhythmia; melanosis coli with chronic use.

Management

Discontinue; correct fluid/electrolyte imbalance; consider potassium supplementation.

Adverse Effects

Cramping abdominal painUrgency / diarrheaYellow-brown to red urine discoloration (harmless)Electrolyte disturbance with prolonged useMelanosis coli (chronic use)

CYP Metabolism

Emodin is a CYP3A4, CYP1A2 and CYP2C9 inhibitor in vitro; clinical relevance uncertain. Stimulant laxatives reduce transit time and can reduce absorption of co-administered oral drugs.

swap_horiz Interactions

Warfarin

Increased Effect high

Class: Anticoagulant (vitamin K antagonist)

Mechanism

Rhubarb acts as a stimulant laxative (anthraquinones rhein, emodin, aloe-emodin, chrysophanol). Diarrhea reduces vitamin K absorption and alters gut flora, increasing warfarin's anticoagulant effect. Anthraquinones also show intrinsic antiplatelet activity.

Clinical Guidance

Avoid chronic rhubarb laxative use in anticoagulated patients. If used short-term, monitor INR and watch for bleeding. Discontinue if diarrhea occurs.

menu_book
Evidence Source Natural Medicines Comprehensive Database: Rhubarb. TRC Healthcare; 2024 View source open_in_new

Digoxin

Increased Effect high

Class: Cardiac glycoside

Mechanism

Chronic stimulant laxative use (including rhubarb) causes potassium depletion. Hypokalemia potentiates digoxin binding to the Na+/K+-ATPase, increasing risk of digoxin toxicity (arrhythmia, nausea, visual changes) at therapeutic serum levels.

Clinical Guidance

Avoid chronic rhubarb use in patients on digoxin. Check serum potassium and digoxin level within 1-2 weeks of initiation. Replace potassium if needed.

menu_book
Evidence Source Memorial Sloan Kettering Cancer Center. Rhubarb monograph. Updated 2024 View source open_in_new

Loop and thiazide diuretics (furosemide, hydrochlorothiazide)

Caution moderate

Class: Diuretic

Mechanism

Stimulant-laxative-induced GI potassium loss combined with kaliuretic diuretics can precipitate severe hypokalemia, leading to arrhythmias, muscle weakness, and metabolic alkalosis.

Clinical Guidance

Avoid chronic combined use. Monitor serum potassium and magnesium regularly. Consider potassium-sparing diuretic or potassium supplementation.

menu_book
Evidence Source WebMD: Rhubarb monograph. Therapeutic Research Center; 2024 View source open_in_new

Corticosteroids (prednisone, hydrocortisone)

Caution moderate

Class: Glucocorticoid

Mechanism

Both anthraquinone laxatives and corticosteroids lower serum potassium. Additive hypokalemia may cause cardiac arrhythmias and muscle weakness, especially in high-dose or long-term steroid use.

Clinical Guidance

Monitor electrolytes when combined. Replace potassium proactively. Prefer bulk-forming or osmotic laxative alternatives.

menu_book
Evidence Source WebMD: Rhubarb monograph. Therapeutic Research Center; 2024 View source open_in_new

Cyclosporine

Decreased Effect high

Class: Immunosuppressant (calcineurin inhibitor)

Mechanism

In rats, rhubarb significantly decreased systemic exposure (AUC) of cyclosporine, which is metabolized by CYP3A4 and effluxed by P-glycoprotein. Rhubarb modulates both pathways and its laxative action reduces absorption time.

Clinical Guidance

Avoid rhubarb in transplant patients on cyclosporine. Monitor cyclosporine trough levels closely if exposure occurs; consider dose increase if levels fall.

menu_book
Evidence Source Yu CP et al. Xenobiotica 2016;46(8):677-682 View source open_in_new

Methotrexate

Increased Effect moderate

Class: Antineoplastic / Antirheumatic (antimetabolite)

Mechanism

In rats, rhubarb co-administration altered methotrexate pharmacokinetics, likely via anthraquinone inhibition of organic anion transporters (OAT1/OAT3) that clear methotrexate renally, elevating systemic exposure.

Clinical Guidance

Avoid concurrent use in patients on methotrexate for cancer or autoimmune disease. Monitor LFTs, creatinine, and CBC; watch for mucositis and myelosuppression.

menu_book
Evidence Source Shia CS et al. Am J Chin Med 2013;41(6):1427-1438 View source open_in_new

Oral medications (general)

Decreased Effect low

Class: All oral drugs

Mechanism

Rhubarb is a stimulant laxative that reduces gastrointestinal transit time. Rapid transit can reduce absorption of orally administered medications, particularly those with slow dissolution or absorption in the small intestine.

Clinical Guidance

Take oral medications at least 2 hours before or after rhubarb products. Monitor response to chronic oral therapies if rhubarb use is ongoing.

menu_book
Evidence Source Drugs.com: Rhubarb monograph. 2024 View source open_in_new

Other stimulant laxatives (senna, bisacodyl, cascara)

Synergistic high

Class: Stimulant laxative

Mechanism

Additive anthraquinone/diphenylmethane laxative effects can produce severe diarrhea, dehydration, electrolyte derangement (hypokalemia, hypomagnesemia), and melanosis coli with chronic use.

Clinical Guidance

Do not combine stimulant laxatives. Limit rhubarb use to short courses (< 1-2 weeks). Use osmotic or bulk-forming alternatives for chronic constipation.

menu_book
Evidence Source WebMD: Rhubarb monograph. Therapeutic Research Center; 2024 View source open_in_new

hub Combinations

info

Synergistic pairings can enhance therapeutic outcomes, while knowing suitable substitutes helps when specific herbs are unavailable or contraindicated.

receipt_long

Classical Formulas

4
Rationale

Classic pairing in Da Huang Fu Zi Tang for Cold accumulation with constipation; warms while purging.

Clinical Evidence

Empirical TCM use since Han dynasty.

link Bensky D et al. Formulas & Strategies, 2nd ed. 2009
Chinese Skullcap
Traditional Use
Rationale

Triad with Coptis in San Huang Xie Xin Tang for Heat with bleeding; anti-inflammatory and hemostatic synergy.

Clinical Evidence

Documented use in Damp-Heat syndromes.

link Bensky D et al. Formulas & Strategies, 2nd ed. 2009
Goldthread
Traditional Use
Rationale

Pair in San Huang Xie Xin Tang with Scutellaria baicalensis for heat with upper GI bleeding, agitation, and hypertension.

Clinical Evidence

Used in TCM for acute hypertension and bleeding disorders.

link Bensky D et al. Formulas & Strategies, 2nd ed. 2009
Mirabilite (Mang Xiao)
Moderate Evidence
Rationale

Pair in Da Cheng Qi Tang; Mirabilite softens hardness, Da Huang purges — the core purgative combination.

Clinical Evidence

Used acutely in hospital TCM settings for ileus and severe constipation.

swap_horiz

Possible Substitutes

1
Senna
Strong Evidence
Rationale

Both are anthraquinone stimulant laxatives with nearly identical mechanisms; Senna is preferred in Western practice for short-term constipation.

Clinical Evidence

Pharmacologically equivalent mechanism; comparative efficacy data.

science Studies

search

Constipation Mitigation by Rhubarb Extract in Middle-Aged Adults Is Linked to Gut Microbiome Modulation: A Double-Blind Randomized Placebo-Controlled Trial

RCT
2022 |Neyrinck AM, Rodriguez J, Taminiau B, et al. Int J Mol Sci. 2022;23(23):14685

This double-blind, placebo-controlled RCT randomized middle-aged adults (95% women, avg. 58 years) with constipation into three groups: rhubarb extract at 12.5 mg/day rhein, 25 mg/day rhein, or placebo (maltodextrin) for 30 days. Both rhubarb doses significantly improved stool frequency, consistency, and perceived transit speed compared to placebo. Rhubarb extract supplementation increased Lachnospiraceae (specifically Roseburia and Agathobacter) abundance and short-chain fatty acid (SCFA) production. Fecal Lachnospiraceae and SCFA levels correlated positively with stool consistency improvements, suggesting gut microbiome modulation underlies the laxative benefit.

ConstipationDigestive Disorders
laxativegut microbiome modulationprebioticSCFA production
View source open_in_new

Meta-Analysis of Efficacy of Rhubarb Combined With Early Enteral Nutrition for the Treatment of Severe Acute Pancreatitis

Meta-Analysis
2020 |Chen X, Yang K, Jing G, Yang J, Li K. JPEN J Parenter Enteral Nutr. 2020;44(6):1066-1078

This meta-analysis pooled 11 randomized controlled trials comprising 724 patients with severe acute pancreatitis (SAP) to evaluate rhubarb combined with early enteral nutrition versus EEN alone. Rhubarb plus EEN significantly reduced hospital stay (MD -4.49 days), ICU stay (MD -2.82 days), abdominal pain duration (MD -2.20 days), and distension duration (MD -2.31 days) compared to EEN alone. Additionally, white blood cell counts and CRP were significantly lower in the rhubarb group. Hospitalization costs were also substantially reduced. These data strongly support rhubarb as a beneficial adjunct in SAP management.

Acute pancreatitisInflammation
anti-inflammatorygut motilityintestinal barrier protection
View source open_in_new

medication Dosing

decoction

Dose Range

3-15 g dried root (purgative); 1-3 g (digestive bitter)

Frequency

1x/day at bedtime for laxative effect

Notes

Add Da Huang in the last 5 minutes of decoction (hou xia) to preserve purgative anthraquinones; prolonged cooking destroys them.

tincture

Dose Range

0.5-2 mL (1:5, 60% ethanol)

Frequency

1-2x/day

Notes

Low doses for bitter tonic effect; short-term only for constipation.

capsule

Dose Range

20-30 mg hydroxyanthracene derivatives (calculated as rhein)

Frequency

1x/day at bedtime

Notes

EMA maximum; do not use longer than 1-2 weeks without medical supervision.

smart_toy

Disclaimer: This information is largely AI-generated and reviewed by human experts at Evara Health. It is intended for educational and clinical reference purposes only and should not replace professional medical advice.

© 2026 Evara Health. All rights reserved.

Clinical Action Center

Export data for clinical use or patient education