Wormwood

Asteraceae

Artemisia absinthium

Also known as: Absinthium, Common Wormwood, Green Ginger

Pregnancy X
Lactation X

clinical_notes Clinical Summary

Wormwood (Artemisia absinthium) is a bitter aromatic herb of Mediterranean origin whose thujone-containing essential oil is infamous as the active principle of absinthe.

Clinically, low-thujone preparations are used as bitter digestives, carminatives, and anthelmintics, with a notable 2007 double-blind RCT showing steroid-sparing effects in Crohn's disease.

Because of thujone's abortifacient, convulsant, and neurotoxic properties, it is absolutely contraindicated in pregnancy, lactation, and seizure disorders; aqueous extracts at controlled doses remain the safer clinical form.

Pregnancy Safety

X

Absolutely contraindicated in pregnancy. Thujone is a known abortifacient and neurotoxin. Australian TGA recalled Artemisia absinthium products over pregnancy risks in 2021.

Lactation Safety

X

Contraindicated during breastfeeding. Thujone is neurotoxic and transfers into breast milk.

warning Contraindications

  • Pregnancy (contraindicated)
    Theoretical
  • Breastfeeding (contraindicated)
    Theoretical
  • Seizure disorder / Epilepsy (contraindicated)
    Theoretical
  • Peptic ulcer disease / Gastric hyperacidity (avoid)
    Clinically Proven
  • Asteraceae/Compositae allergy (avoid)
    Clinically Proven

vital_signs Clinical Profile

Primary Indications

  • check_circle intestinal parasites
  • check_circle dyspepsia
  • check_circle loss of appetite
  • check_circle Crohn's disease
  • check_circle biliary insufficiency
  • check_circle IgA nephropathy

Therapeutic Actions

bitter tonicanthelminticcholereticcarminativeanti-inflammatoryantimicrobialantimalarial

System Affinities

  • check_circle digestive system
  • check_circle liver
  • check_circle gallbladder
  • check_circle intestines

labs Active Constituents

absinthin

anabsinthin

thujone

sesquiterpene lactones

chamazulene

phenolic acids

flavonoids

essential oil

history_edu Traditional Use

Traditional Chinese Medicine (TCM)

Chinese Name

苦艾 (Ku Ai)

Properties

Nature: cool

bitterpungent
Meridians / Channels
LiverSpleenStomach
TCM Indications
  • damp-heat dysentery
  • food stagnation
  • parasitic infestation
  • summer-heat
Zang-Fu Organ Patterns
Spleen Damp-HeatFood Stagnation with Damp-Heat
Notes

Used in folk Chinese medicine (distinct from common mugwort Ai Ye / Artemisia argyi) — sometimes for bacillary dysentery externally.

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Traditional Uses Across Healing Systems

While many herbs lack controlled clinical trials, centuries of traditional practice across cultures provide valuable insight into their therapeutic applications.

Western Herbal Europe
Since antiquity; featured in Ebers Papyrus (1550 BCE)

Bitter digestive tonic for dyspepsia, anorexia, biliary insufficiency; vermifuge for roundworms and pinworms.

Approved by German Commission E for loss of appetite and dyspeptic complaints.

Unani Middle East, South Asia
Medieval Islamic medicine onward

Afsanteen — used for hepatic disorders, fever, and as anthelmintic.

Classified as hot and dry.

TCM China
Traditional folk use

External poultice for tendon inflammation; fresh or dried application for acute bacillary dysentery.

Distinct from Ai Ye (Artemisia argyi) in mainstream TCM practice.

spa Parts Used

aerial parts

Constituents
absinthinanabsinthinthujonechamazuleneflavonoidsessential oil
Indications
  • dyspepsia
  • anorexia
  • parasites
  • Crohn's disease
Preparation

Aerial parts (leaves and flowering tops) harvested at flowering. Aqueous extracts (teas) have markedly lower thujone content than essential oil or alcoholic extracts.

shield Safety

Contraindications — Evidence Basis

Pregnancy
contraindicated Theoretical

Thujone is an abortifacient and neurotoxic; Australian TGA recalled Artemisia absinthium products in 2021 over pregnancy risk.

Breastfeeding
contraindicated Theoretical

Thujone passes into breast milk and is neurotoxic to infants.

Seizure disorder / Epilepsy
contraindicated Theoretical

Thujone is a GABA-A receptor antagonist and can provoke seizures; 13-week rat study showed convulsions at 25 mg/kg/day thujone.

Peptic ulcer disease / Gastric hyperacidity
avoid Clinically Proven

Bitter principles stimulate gastric acid secretion and may aggravate ulcer disease.

Asteraceae/Compositae allergy
avoid Clinically Proven

Cross-reactivity with ragweed, mugwort; reports of rhinitis, dermatitis.

monitoring

Monitoring Parameters

Monitor during use, especially with prolonged or high-dose therapy.

Liver enzymes (ALT, AST)
Baseline and every 4-6 weeks during therapeutic use

Thujone is hepatotoxic at high/chronic doses; essential oil particularly concerning

flagThreshold: ALT/AST >3x ULN: discontinue and reassess

Renal function (creatinine, BUN)
Baseline and every 4-6 weeks

Thujone-containing preparations have been associated with acute kidney injury

flagThreshold: Creatinine rise >30% from baseline: discontinue

Toxicity

Toxic Dose

Essential oil toxic at doses >15mL; thujone LD50 in rats ~120 mg/kg oral; convulsions seen at 25 mg/kg/day thujone chronically.

Symptoms

Absinthism syndrome: convulsions, hallucinations, tremors, insomnia, stupor, vomiting, diarrhea, urinary retention, renal injury, hepatotoxicity.

Management

Discontinue immediately; benzodiazepines for seizures; supportive care; activated charcoal if recent ingestion; renal and hepatic monitoring.

Adverse Effects

nauseavomitingheadachedizzinessallergic dermatitis/rhinitisseizures (high dose)

CYP Metabolism

Thujones detoxified by CYP2A6, CYP2B6, and CYP3A4 to 7-hydroxythujone. Individuals with CYP2A6 polymorphisms may have prolonged thujone exposure. Avoid co-administration with CYP2A6/3A4 inhibitors.

swap_horiz Interactions

Phenobarbital

Antagonistic high

Class: Barbiturate anticonvulsant / GABA-A modulator

Mechanism

α-Thujone is a rapidly acting antagonist of the GABA-gated chloride channel, producing excitation and seizures; it pharmacodynamically opposes the GABA-enhancing action of barbiturates and benzodiazepines, potentially reducing seizure threshold.

Clinical Guidance

Contraindicated in epilepsy and in patients taking GABAergic anticonvulsants (phenobarbital, primidone, clonazepam, diazepam). Use only thujone-free (<0.35 mg/kg) preparations in this population.

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Evidence Source Höld KM et al. Alpha-thujone (the active component of absinthe): gamma-aminobutyric acid type A receptor modulation and metabolic detoxification. Proc Natl Acad Sci USA 2000;97(8):3826-3831 View source open_in_new

Itraconazole

Increased Effect high

Class: Azole antifungal (CYP3A4 inhibitor)

Mechanism

α-Thujone undergoes 7- and 4-hydroxylation primarily by CYP2A6 with CYP3A4 and CYP2B6 as minor pathways. Strong CYP3A4 inhibitors (itraconazole, ketoconazole, ritonavir, clarithromycin) slow thujone detoxification and increase neurotoxic exposure, particularly in CYP2A6 poor-metabolisers.

Clinical Guidance

Avoid wormwood essential-oil and high-dose tincture preparations with strong CYP3A4 inhibitors. Thujone-free herbal preparations pose no such risk.

menu_book
Evidence Source Abass K et al. Metabolism of α-thujone in human hepatic preparations in vitro. Xenobiotica 2011;41(2):101-111 View source open_in_new

Methoxsalen (8-MOP)

Increased Effect high

Class: CYP2A6 inhibitor / photochemotherapy

Mechanism

CYP2A6 performs 70–80% of α-thujone 4- and 7-hydroxylation in human liver microsomes. Methoxsalen, a potent CYP2A6 inhibitor, blocks thujone detoxification, prolonging GABA-antagonist effect and raising seizure risk.

Clinical Guidance

Avoid thujone-containing wormwood preparations with methoxsalen, pilocarpine, or other CYP2A6 inhibitors; recommend processed or thujone-limited (EMA <3 mg/day) preparations for ≤2 weeks only.

menu_book
Evidence Source European Medicines Agency. Assessment report on Artemisia absinthium L., herba. EMA/HMPC/751484/2016 View source open_in_new

Warfarin

Increased Effect high

Class: Anticoagulant

Mechanism

Case report documented probable warfarin-wormwood interaction with elevated INR and gastrointestinal bleeding; flavonoids and sesquiterpenes may inhibit CYP2C9-mediated S-warfarin metabolism and/or hepatic clearance.

Clinical Guidance

Avoid concurrent use. If wormwood is being used, check INR at day 3, 7, and 14 after initiation and watch for GI bleeding; dose-reduce warfarin if INR rises.

menu_book
Evidence Source Açıkgöz SK et al. A probable interaction between warfarin and Artemisia absinthium: a case report. Blood Coagul Fibrinolysis 2013;24(6):669-670 View source open_in_new

Valproic acid

Antagonistic high

Class: Anticonvulsant

Mechanism

Thujone-mediated GABA-A antagonism lowers seizure threshold and can precipitate convulsions despite therapeutic valproate levels; essential-oil wormwood preparations have caused tonic-clonic seizures in case reports.

Clinical Guidance

Contraindicated in patients with seizure disorders on any anticonvulsant. Advise epilepsy patients that absinthe-style wormwood preparations must be avoided.

menu_book
Evidence Source Weisbord SD, Soule JB, Kimmel PL. Poison on line—acute renal failure caused by oil of wormwood purchased through the Internet. N Engl J Med 1997;337(12):825-827 View source open_in_new

hub Combinations

info

Synergistic pairings can enhance therapeutic outcomes, while knowing suitable substitutes helps when specific herbs are unavailable or contraindicated.

receipt_long

Classical Formulas

2
Black Walnut
Traditional Use
Rationale

Classic parasite cleanse triad with clove — broad-spectrum antiparasitic synergy targeting different life-cycle stages.

Clinical Evidence

Traditional combination; limited formal RCT evidence.

link Clark HR. The Cure for All Diseases, 1995
Clove
Traditional Use
Rationale

Eugenol in clove destroys parasite eggs while wormwood targets adult stages.

Clinical Evidence

Traditional antiparasitic combination.

link Clark HR. The Cure for All Diseases, 1995
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Possible Substitutes

1
Mugwort
Traditional Use
Rationale

Mugwort (Artemisia vulgaris) has gentler bitter and emmenagogue action — sometimes used as a milder substitute in digestive and menstrual formulas.

Clinical Evidence

Traditional Western practice.

link Mills & Bone, Principles and Practice of Phytotherapy, 2013
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Synergistic Combinations

2
Fennel
Traditional Use
Rationale

Fennel's carminative action offsets wormwood's potential GI irritation while complementing digestive support.

Clinical Evidence

Traditional European digestive formulation.

link British Herbal Pharmacopoeia, 1983
Gentian
Traditional Use
Rationale

Both are potent bitters; synergistic stimulation of digestive secretions with complementary gentle and intense bitter profiles.

Clinical Evidence

Traditional European bitter formulation (featured in Swedish Bitters).

link Hoffmann D. Medical Herbalism, 2003

science Studies

search

Topical Effects of Artemisia Absinthium Ointment and Liniment in Comparison with Piroxicam Gel in Patients with Knee Joint Osteoarthritis: A Randomized Double-Blind Controlled Trial

RCT
2018 |Zargaran A, Borhani-Haghighi A, Faridi P, et al. Iran J Med Sci. 2018;43(1):14-21

This randomised double-blind trial enrolled 90 patients (aged 30–70) with primary knee osteoarthritis and assigned them to topical Artemisia absinthium ointment 3% (AAO), A. absinthium liniment 3% (AAL), or piroxicam gel (PG) applied three times daily for 4 weeks. Both wormwood formulations produced meaningful reductions in pain and improved functional status. The AA ointment group showed beneficial effects comparable to piroxicam gel in relieving OA symptoms. These findings support the traditional use of A. absinthium as a topical anti-inflammatory agent for musculoskeletal pain.

anti-inflammatoryanalgesic
View source open_in_new

Wormwood (Artemisia absinthium) for poorly responsive early-stage IgA nephropathy: a pilot uncontrolled trial

Case Study
2010 |Krebs S, Omer B, Djafarian K. J Nephrol. 2010;23(6):694-700

This pilot uncontrolled trial enrolled 10 patients with biopsy-proven IgA nephropathy who had proteinuria >500 mg/day despite at least 3 months of dual renin-angiotensin system (RAS) blockade. Patients received 1.8 g/day of thujone-free wormwood preparation for 6 months as a supplement, while continuing RAS blockade. Proteinuria decreased and kidney function parameters showed improvement in several patients. Given the known role of TNF-alpha in IgA nephropathy and wormwood's TNF-alpha-suppressing properties, the results suggest a potential role for A. absinthium as adjunctive therapy in this autoimmune kidney disease, warranting further controlled investigation.

anti-inflammatoryTNF-alpha inhibitionimmunomodulatory
View source open_in_new

medication Dosing

tea

Dose Range

1-1.5 g dried herb in 150 mL boiling water

Frequency

TID before meals

Notes

Maximum 3g/day. Short-term use only (max 4 weeks). Aqueous extract has low thujone content.

tincture

Dose Range

1-4 mL (1:5 in 40% ethanol)

Frequency

TID before meals

Notes

Short-term use; thujone content higher in alcoholic extract. Final product should contain <6 mg thujone/day.

capsule

Dose Range

500-1500 mg dried herb/day

Frequency

divided TID

Notes

Steroid-sparing Crohn's study used SedaCrohn 3x500 mg/day with total daily thujone <6 mg.

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Disclaimer: This information is largely AI-generated and reviewed by human experts at Evara Health. It is intended for educational and clinical reference purposes only and should not replace professional medical advice.

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